Papers：2017

No.118Synthetic Study toward Total Synthesis of (±)-Germine: Synthesis of (±)-4-Methylenegermine

Stork, G.; Yamashita, A.; Hanson, R. M.; Phan, L.; Phillips, E.; Dubé, D.; Bos, P. H.; Clark, A. J.; Gough, M.; Grrenlee, M. L.; Jiang, Y.; Jones, K.; Kitamura, M.; Leonard, J.; Liu, T.; Parsons, P. J.; Venkatesan, A. M. Org. Lett. 2017, 19, 5150–5153.

No.117Modular Construction of Protected 1,2/1,3-Diols, -Amino Alcohols, and -Diamines via Catalytic Asymmetric Dehydrative Allylation: An Application to Synthesis of Sphingosine

Tanaka, S.; Gunasekar, R.; Tanaka, T.; Iyoda, Y.; Suzuki, Y.; Kitamura, M. J. Org. Chem. 2017, 82, 9160–9170.

No.116Synthetic analogs of a protozoan glycolipid designed to combat intracellular Leishmania infection

Choy, S. L.; Bernin, H.; Aiba, T.; Bifeld, E.; Lender, S. C.; Mühlenpfordt, M.; Noll, J.; Eick, J.; Marggra, C.; Niss, H.; Roldán, N. G.; Tanaka, S.; Kitamura, M.; Fukase, K.; Clos, J.; Tannich, E.; Fujimoto, Y.; Lotter, H. Sci. Rep. 2017, 7, 9472 (DOI:10.1038/s41598-017-09894-8).

No.115π-Allyl Donicity Switch in Catalytic Asymmetric Allylation: Usability of a Robust and Feasible Allyl Methyl Ether

Suzuki, Y.; Iwase, S.; Hashimoto, K.; Tanaka, S.; Kitamura, M. Chem. Lett. 2017, 46, 1308–1310.

(Editor’s Choice)

No.114Synthesis and biological evaluation of chemokine receptor ligands with 2-benzazepine scaffold

Thum, S.; Kokornaczyk, A. K.; Seki, T.; Maria, M. D.; Zacarias, N. V. O.; Vries, H.; Weiss, C.; Koch, M.; Schepmann, D.; Kitamura, M.; Tschammer, N.; Heitman, L. H.; Junker, A.; Wünsch, B. Eur. J. Med. Chem. 2017, 135, 401–413.

No.113Do GluN2B subunit containing NMDA receptors tolerate a fluorine atom in the phenylalkyl side chain?

Shuto, Y.; Thum, S.; Temme, L.; Schepmann, D.; Kitamura, M.; Wünsch, B. Med. Chem. Commun. 2017, 8, 975–981.

No.112Enantio- and Diastereoselective Dehydrative “One-Step” Construction of Spirocarbocycles via a Ru/H+-Catalyzed Tsuji-Trost Approach

Suzuki, Y.; Vatmurge, N.; Tanaka, S.; Kitamura, M. Chem. Asian J. 2017, 12, 633–637.